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Takashi Kobunai Selected Research

Trifluridine (Viroptic)

10/2019CD44/CD133-Positive Colorectal Cancer Stem Cells are Sensitive to Trifluridine Exposure.
7/2019ChIP-seq Analysis to Explore DNA Replication Profile in Trifluridine-treated Human Colorectal Cancer Cells In Vitro.
10/2018Thymidine Kinase 1 Loss Confers Trifluridine Resistance without Affecting 5-Fluorouracil Metabolism and Cytotoxicity.
12/2017Improved chemoradiation treatment using trifluridine in human colorectal cancer cells in vitro.
8/2017MicroRNA profiles involved in trifluridine resistance.

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Takashi Kobunai Research Topics

Disease

21Colorectal Neoplasms (Colorectal Cancer)
01/2020 - 01/2007
19Neoplasms (Cancer)
01/2020 - 09/2006
5Rectal Neoplasms (Rectal Cancer)
12/2017 - 08/2008
4Ulcerative Colitis
01/2020 - 01/2007
4Stomach Neoplasms (Stomach Cancer)
03/2018 - 11/2011
4Colonic Neoplasms (Colon Cancer)
03/2016 - 01/2008
1Carcinogenesis
07/2017
1Adenocarcinoma
07/2017
1Body Weight (Weight, Body)
01/2017
1Esophageal Squamous Cell Carcinoma
01/2015
1Non-Small-Cell Lung Carcinoma (Carcinoma, Non-Small Cell Lung)
05/2012
1Breast Neoplasms (Breast Cancer)
05/2012
1Body Weight Changes
05/2012
1Prostatic Neoplasms (Prostate Cancer)
12/2009
1Lymphatic Metastasis
12/2009

Drug/Important Bio-Agent (IBA)

13Fluorouracil (Carac)FDA LinkGeneric
10/2018 - 03/2007
8DNA (Deoxyribonucleic Acid)IBA
01/2020 - 10/2006
5Trifluridine (Viroptic)FDA LinkGeneric
10/2019 - 08/2017
4trifluridine tipiracil drug combinationIBA
07/2019 - 01/2017
4Leucovorin (Folinic Acid)FDA Link
03/2016 - 01/2008
4RNA-Directed DNA Polymerase (Reverse Transcriptase)IBA
01/2014 - 07/2010
3Pharmaceutical PreparationsIBA
10/2018 - 01/2015
2Mitochondrial DNA (mtDNA)IBA
01/2020 - 07/2017
2Antineoplastic Agents (Antineoplastics)IBA
07/2019 - 08/2017
2Thymidylate SynthaseIBA
03/2018 - 08/2011
2Monoclonal AntibodiesIBA
01/2017 - 11/2011
2titanium silicide (TS-1)IBA
03/2016 - 09/2006
2Dihydrouracil Dehydrogenase (NADP) (Dihydropyrimidine Dehydrogenase)IBA
01/2015 - 03/2007
2Oxaliplatin (Eloxatin)FDA LinkGeneric
07/2012 - 06/2011
2Vascular Endothelial Growth Factor A (Vascular Endothelial Growth Factor)IBA
05/2012 - 08/2011
2Cetuximab (Erbitux)FDA Link
05/2012 - 11/2011
2Bevacizumab (Avastin)FDA Link
05/2012 - 08/2011
2Messenger RNA (mRNA)IBA
01/2011 - 11/2007
1tipiracilIBA
10/2019
1NucleosidesIBA
10/2018
1Nonsense Codon (Nonsense Mutation)IBA
10/2018
1thymidine kinase 1IBA
10/2018
1Ribosomal Protein S6 Kinases (S6 Kinase)IBA
01/2017
12- (1H- indazol- 4- yl)- 6- (4- methanesulfonylpiperazin- 1- ylmethyl)- 4- morpholin- 4- ylthieno(3,2- d)pyrimidineIBA
01/2017
1UracilIBA
03/2016
1TegafurIBA
03/2016
1S-1 plus cisplatinIBA
01/2016
1Receptor Protein-Tyrosine Kinases (Tyrosine Kinase Receptors)IBA
01/2016
1Biomarkers (Surrogate Marker)IBA
11/2012
1Capecitabine (Xeloda)FDA Link
07/2012
1Sunitinib (Sutent)FDA Link
05/2012
1Erlotinib Hydrochloride (CP 358,774)FDA Link
05/2012
1AntibodiesIBA
05/2012
1Tyrosine Kinase InhibitorsIBA
05/2012
1Sorafenib (BAY 43-9006)FDA Link
05/2012
1ErbB Receptors (EGF Receptor)IBA
11/2011
1ProdrugsIBA
11/2011
1Calcibiotic Root Canal SealerIBA
09/2011
1Tissue Inhibitor of Metalloproteinase-3IBA
08/2011
125-Hydroxyvitamin D3 1-alpha-Hydroxylase (25 Hydroxyvitamin D3 1 alpha Hydroxylase)IBA
06/2011
1Peptide Nucleic AcidsIBA
04/2010
1Glycoproteins (Glycoprotein)IBA
12/2009
1AntimetabolitesIBA
02/2008
1Methylenetetrahydrofolate Reductase (NADPH2) (Methylenetetrahydrofolate Reductase)IBA
02/2008
1pyrimidineIBA
02/2008
1Folic Acid (Vitamin M)FDA LinkGeneric
01/2008
1Orotate PhosphoribosyltransferaseIBA
11/2007
1A-Form DNA (A-DNA)IBA
01/2007

Therapy/Procedure

8Therapeutics
10/2019 - 01/2009
6Drug Therapy (Chemotherapy)
10/2019 - 01/2008
4Chemoradiotherapy
12/2017 - 08/2008
3Radiotherapy
12/2017 - 12/2011
2Adjuvant Chemotherapy
03/2016 - 11/2012
2Combination Drug Therapy (Combination Chemotherapy)
07/2012 - 11/2011
2Lymph Node Excision (Lymph Node Dissection)
12/2009 - 08/2008
1Aftercare (After-Treatment)
01/2017
1Ligation
02/2008